Pharmaceutics (ISSN 1999-4923) is an open access journal which provides an advanced forum for the science and technology of pharmaceutics and biopharmaceutics. It publishes reviews, regular research papers, communications, and short notes. Covered topics include pharmacokinetics, toxicokinetics, pharmacodynamics, pharmacogenetics and pharmacogenomics, and pharmaceutical formulation. Our aim is to encourage scientists to publish their experimental and theoretical details in as much detail as possible. There is no restriction on the length of the papers. The full experimental details must be provided so that the results can be reproduced.
《药剂学》(ISSN 1999-4923)是一本开放获取期刊,为药剂学和生物药剂学的科学和技术提供了一个先进的论坛。它发表评论、定期研究论文、通信和简短的笔记。涵盖的主题包括药代动力学、毒代动力学、药效学、药物遗传学和药物基因组学以及药物制剂。我们的目标是鼓励科学家尽可能详细地发表他们的实验和理论细节。论文的长度没有限制。必须提供完整的实验细节,以便重现结果。
Intestinal Permeation Enhancers for Oral Delivery of Macromolecules: A Comparison between Salcaprozate Sodium (SNAC) and Sodium Caprate (C10)
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11020078
Polymeric Mesoporous Silica Nanoparticles for Enhanced Delivery of 5-Fluorouracil In Vitro
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11060288
Protein Corona Fingerprints of Liposomes: New Opportunities for Targeted Drug Delivery and Early Detection in Pancreatic Cancer
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11010031
Nanoconjugation and Encapsulation Strategies for Improving Drug Delivery and Therapeutic Efficacy of Poorly Water-Soluble Drugs
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070325
Penetration Enhancers in Ocular Drug Delivery
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070321
Established and Emerging Strategies for Drug Delivery Across the Blood-Brain Barrier in Brain Cancer
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11050245
Enhanced Oral Bioavailability of Celecoxib Nanocrystalline Solid Dispersion based on Wet Media Milling Technique: Formulation, Optimization and In Vitro/In Vivo Evaluation
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070328
Development and Characterization of the Solvent-Assisted Active Loading Technology (SALT) for Liposomal Loading of Poorly Water-Soluble Compounds
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11090465
Formulation Strategies to Improve Nose-to-Brain Delivery of Donepezil
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11020064
Impact of Processing Parameters on the Quality of Pharmaceutical Solid Dosage Forms Produced by Fused Deposition Modeling (FDM)
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11120633
Systemic Design and Evaluation of Ticagrelor-Loaded Nanostructured Lipid Carriers for Enhancing Bioavailability and Antiplatelet Activity
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11050222
The Self-Assembly Phenomenon of Poloxamers and Its Effect on the Dissolution of a Poorly Soluble Drug from Solid Dispersions Obtained by Solvent Methods
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11030130
Computational Approaches in Theranostics: Mining and Predicting Cancer Data
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11030119
Mechanistic Evaluation of Enhanced Curcumin Delivery through Human Skin In Vitro from Optimised Nanoemulsion Formulations Fabricated with Different Penetration Enhancers
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11120639
Repurposing Butenafine as An Oral Nanomedicine for Visceral Leishmaniasis
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070353
Comparison of Target Features for Predicting Drug-Target Interactions by Deep Neural Network Based on Large-Scale Drug-Induced Transcriptome Data
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11080377
Investigation of Dissolution Mechanism and Release Kinetics of Poorly Water-Soluble Tadalafil from Amorphous Solid Dispersions Prepared by Various Methods
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11080383
The Impact of Solvent Selection: Strategies to Guide the Manufacturing of Liposomes Using Microfluidics
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11120653
1,4-Dihydropyridine Antihypertensive Drugs: Recent Advances in Photostabilization Strategies
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11020085
What Drives Innovation: The Canadian Touch on Liposomal Therapeutics
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11030124
Oxaliplatin–Biomimetic Magnetic Nanoparticle Assemblies for Colon Cancer-Targeted Chemotherapy: An In Vitro Study
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11080395
Synthesis and Preclinical Evaluation of Radio-Iodinated GRPR/PSMA Bispecific Heterodimers for the Theranostics Application in Prostate Cancer
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070358
Evaluation of Sucrose Laurate as an Intestinal Permeation Enhancer for Macromolecules: Ex Vivo and In Vivo Studies
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11110565
Novel Formulations of C-Peptide with Long-Acting Therapeutic Potential for Treatment of Diabetic Complications
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11010027
Potential Use of the Maillard Reaction for Pharmaceutical Applications: Gastric and Intestinal Controlled Release Alginate-Albumin Beads
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11020083
Targeting Cell Adhesion Molecules via Carbonate Apatite-Mediated Delivery of Specific siRNAs to Breast Cancer Cells In Vitro and In Vivo
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070309
Evolution from Covalent to Self-Assembled PAMAM-Based Dendrimers as Nanovectors for siRNA Delivery in Cancer by Coupled in Silico-Experimental Studies. Part II: Self-Assembled siRNA Nanocarriers
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070324
Comprehensive Analysis of the Safety Profile of a Single-Stranded RNA Nano-Structure Adjuvant
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11090464
Be Aggressive! Amorphous Excipients Enabling Single-Step Freeze-Drying of Monoclonal Antibody Formulations
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11110616
Silicon Nanotubes as Potential Therapeutic Platforms
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11110571
Gold Nanocage-Incorporated Poly(ε-Caprolactone) (PCL) Fibers for Chemophotothermal Synergistic Cancer Therapy
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11020060
Stabilisation and Growth of Metastable Form II of Fluconazole in Amorphous Solid Dispersions
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics12010012
Pharmaceutical Applications of Hot-Melt Extrusion: Continuous Manufacturing, Twin-Screw Granulations, and 3D Printing
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11050218
Intracellular PD Modelling (PDi) for the Prediction of Clinical Activity of Increased Rifampicin Dosing
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11060278
Mechanically Robust Gastroretentive Drug-Delivery Systems Capable of Controlling Dissolution Behaviors of Coground β-Lapachone
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11060271
Synthesis and Characterization of pH-Sensitive Inulin Conjugate of Isoniazid for Monocyte-Targeted Delivery
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11110555
Antimicrobial Biophotonic Treatment of Ampicillin-Resistant Pseudomonas aeruginosa with Hypericin and Ampicillin Cotreatment Followed by Orange Light
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11120641
β-Cyclodextrin as a Functional Excipient Used for Enhancing the Diminazene Aceturate Bioavailability
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11060295
Nanomedicine against Aβ Aggregation by β–Sheet Breaker Peptide Delivery: In Vitro Evidence
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11110572
Utilizing a Kidney-Targeting Peptide to Improve Renal Deposition of a Pro-Angiogenic Protein Biopolymer
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11100542
Oxytetracycline versus Doxycycline Collagen Sponges Designed as Potential Carrier Supports in Biomedical Applications
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11080363
Montelukast Nanocrystals for Transdermal Delivery with Improved Chemical Stability
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics12010018
Thermosensitive Liposome-Mediated Drug Delivery in Chemotherapy: Mathematical Modelling for Spatio–temporal Drug Distribution and Model-Based Optimisation
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11120637
Metal-Phenolic Network-Coated Hyaluronic Acid Nanoparticles for pH-Responsive Drug Delivery
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11120636
Contribution of Molecular Structure to Self-Assembling and Biological Properties of Bifunctional Lipid-Like 4-(N-Alkylpyridinium)-1,4-Dihydropyridines
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11030115
Supercritical Solvent Impregnation of Different Drugs in Mesoporous Nanostructured ZnO
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11070340
Retinal Pigment Epithelial Cell Line with Fast Differentiation and Improved Barrier Properties
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11080412
A Low-Molecular-Weight Polyethylenimine/pDNA-VEGF Polyplex System Constructed in a One-Pot Manner for Hindlimb Ischemia Therapy
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11040171
Determining Thermal Conductivity of Small Molecule Amorphous Drugs with Modulated Differential Scanning Calorimetry and Vacuum Molding Sample Preparation
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11120670
Extended Release Combination Antibiotic Therapy from a Bone Void Filling Putty for Treatment of Osteomyelitis
来源期刊:PharmaceuticsDOI:10.3390/pharmaceutics11110592